BDBM138515 US8877775, 26::US9073869, 26
SMILES CS(=O)(=O)c1ccc(cc1C#N)-c1ccc(C[C@H](NC(=O)C2NC3CCC2CC3)C#N)c(F)c1
InChI Key InChIKey=TXKVDXAWFGASKU-DQLVKDCISA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 138515
Affinity DataIC50: 27.8nMT: 2°CAssay Description:The recombinant human DPPI was diluted in TAGZyme buffer to 1 U/ml (38.1 ug/ml, respectively), and then activated by mixing in a 1:2 ratio with a Cys...More data for this Ligand-Target Pair
Affinity DataIC50: 27.8nMpH: 6.0 T: 2°CAssay Description:The following buffers were used: MES buffer: 25 mM MES, 50 mM NaCl, 5 mM DTT, adjusted to pH 6.0, containing 0.1% BSA; TAGZyme Buffer: 20 mM NaH2P04,...More data for this Ligand-Target Pair