BDBM142654 US8937068, 30

SMILES Oc1ccc(cc1)-c1cnc2ccc(NC(=S)NCC=C)nc2n1

InChI Key InChIKey=YKMUCILEPVJXKD-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 142654   

LigandPNGBDBM142654(US8937068, 30)
Affinity DataIC50: 370nMAssay Description:The inhibitory effect of the compounds according to the invention was tested on various serine/threonine, tyrosine and lipid kinases in enzymatic ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2015
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Human)
Zentaris

US Patent
LigandPNGBDBM142654(US8937068, 30)
Affinity DataIC50: 392nMAssay Description:The inhibitory effect of the compounds according to the invention was tested on various serine/threonine, tyrosine and lipid kinases in enzymatic ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2015
Entry Details
US Patent

TargetMitogen-activated protein kinase 8/9(Human)
Zentaris

US Patent
LigandPNGBDBM142654(US8937068, 30)
Affinity DataIC50: 2.18E+4nMAssay Description:The inhibitory effect of the compounds according to the invention was tested on various serine/threonine, tyrosine and lipid kinases in enzymatic ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2015
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Zentaris

US Patent
LigandPNGBDBM142654(US8937068, 30)
Affinity DataIC50: 1.00E+5nMAssay Description:The inhibitory effect of the compounds according to the invention was tested on various serine/threonine, tyrosine and lipid kinases in enzymatic ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2015
Entry Details
US Patent