BDBM143117 US9682953, 2.1

SMILES CN(CCCO)c1ccc(NC(=O)c2cn(C)c3c(CN4CC5N(N(CC=C)CC(=O)N5[C@@H](Cc5ccc(O)cc5)C4=O)C(=O)NCc4ccccc4)cccc23)cn1

InChI Key InChIKey=MLOOBNLWEUZTPL-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 143117   

TargetFatty-acid amide hydrolase 1(Human)
Advinus Therapeutics

US Patent
LigandPNGBDBM143117(US9682953, 2.1)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:All reagents were purchased from Sigma-Aldrich unless specified. Human and Rat Fatty Acid Amide Hydrolase (FAAH) genes used in assay have been descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2018
Entry Details
US Patent

TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Advinus Therapeutics

US Patent
LigandPNGBDBM143117(US9682953, 2.1)
Affinity DataIC50: 24nMpH: 7.4 T: 2°CAssay Description:All reagents were purchased from Sigma-Aldrich unless specified. Human and Rat Fatty Acid Amide Hydrolase (FAAH) genes used in assay have been descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2018
Entry Details
US Patent