BDBM151177 BDBM151178::US8987287, 7
SMILES Oc1ccc2C[C@@H]3[C@@H]4CC[C@@]5(C[C@]4(CCN3CC3CC3)c2c1)NC(=O)NC5=O
InChI Key InChIKey=DNESVBVDIIHDKK-REIYTJMXSA-N
Data 3 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 151177
Affinity DataKi: 0.200nM ΔG°: -13.2kcal/molepH: 7.4 T: 25°CAssay Description:Radioligand dose displacement assays used 0.4 nM [3H]-U69,593 (GE Healthcare, Piscataway, N.J.; 40 Ci/mmole) with 15 ug membrane protein (recombinant...More data for this Ligand-Target Pair
Affinity DataKi: 0.230nM ΔG°: -13.1kcal/molepH: 7.4 T: 25°CAssay Description:Radioligand dose displacement assays used 0.4 nM [3H]-U69,593 (GE Healthcare, Piscataway, N.J.; 40 Ci/mmole) with 15 ug membrane protein (recombinant...More data for this Ligand-Target Pair
Affinity DataKi: 8.39nM ΔG°: -11.9kcal/molepH: 7.4 T: 50°CAssay Description:mu-Opioid Receptor Binding Assay Procedures: Radioligand dose-displacement binding assays for mu-opioid receptors used 0.3 nM [3H]-diprenorphine (Per...More data for this Ligand-Target Pair