BDBM151784 US8987445, 220

SMILES CCOC(C)(c1ccc(CN(c2ncc3ccccc3c2C)S(=O)(=O)c2ccc(cc2)C(O)=O)cc1F)C(F)(F)F

InChI Key InChIKey=OIPUEMNDSSUCMT-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 151784   

TargetTransient receptor potential cation channel subfamily M member 8(Human)
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM151784(US8987445, 220)
Affinity DataIC50: 5nMT: 2°CAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+ sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent