BDBM152763 US10023561, Example 127::US9682965, 127

SMILES CO[C@@H]1[C@@H](CC[C@]2(CO2)[C@H]1[C@@]1(C)O[C@@H]1CCC(C)C)OC(=O)N1CC(CCN2CCOCC2)C1

InChI Key InChIKey=INQYUJFIXMFFKL-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 152763   

TargetMethionine aminopeptidase 2(Human)
Zafgen

US Patent
LigandPNGBDBM152763(US9682965, 127 | US10023561, Example 127)
Affinity DataIC50: 275nMpH: 7.4Assay Description:The plate was sealed with a TopSeal A cover and mixed briefly on an orbital mixer at 900 rpm. The plate was incubated for a further 25 minutes at 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2019
Entry Details
US Patent

TargetMethionine aminopeptidase 2(Human)
Zafgen

US Patent
LigandPNGBDBM152763(US9682965, 127 | US10023561, Example 127)
Affinity DataIC50: 275nMpH: 7.4Assay Description:Flag tagged Human recombinant MetAP2 expressed and isolated for use as the enzyme source. 10 mM stock solutions of compounds were prepared in 100% DM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2018
Entry Details
US Patent