BDBM156351 US9018217, (S)-1-{2-[2-(5,7-Dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-ethyl]-4-phenyl-imidazol-1-yl}-propan-2-ol::US9592230, (S)-1-{2-[2-(5,7-Dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-ethyl]-4-phenyl-imidazol-1-yl}-propan-2-ol

SMILES C[C@H](O)Cn1cc(nc1CCc1nc2nc(C)cc(C)n2n1)-c1ccccc1

InChI Key InChIKey=ZWZHAWCKFMTSMU-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 156351   

LigandPNGBDBM156351(US9018217, (S)-1-{2-[2-(5,7-Dimethyl-[1,2,4]triazo...)
Affinity DataIC50: 5.5nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
US Patent

LigandPNGBDBM156351(US9018217, (S)-1-{2-[2-(5,7-Dimethyl-[1,2,4]triazo...)
Affinity DataIC50: 5.5nMAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2019
Entry Details
US Patent