BDBM160981 US9108903, 46
SMILES OCc1ccc(Oc2cc(cc(c2C(=O)Nc2ccc(nc2)C(O)=O)C(F)(F)F)C(F)(F)F)cc1
InChI Key InChIKey=AGFINBANYZVEFJ-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 160981
TargetSodium channel protein type 10 subunit alpha(Rattus norvegicus (Rat))
Vertex Pharmaceuticals
US Patent
Vertex Pharmaceuticals
US Patent
Affinity DataIC50: 66nMAssay Description:Patch clamp electrophysiology was used to assess the efficacy and selectivity of sodium channel blockers in dorsal root ganglion neurons. Rat neurons...More data for this Ligand-Target Pair