BDBM170486 US9085540, 26

SMILES CN1CCN(CC1)c1ccc(Nc2nc(Oc3cccc(NC(=O)C=C)c3)cnc2C(N)=O)cc1

InChI Key InChIKey=YGIBTSMHVRPSJH-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 170486   

TargetEpidermal growth factor receptor(Human)
Astellas Pharma

US Patent
LigandPNGBDBM170486(US9085540, 26)
Affinity DataIC50: 0.920nMAssay Description:The phosphorylation activity on the peptide substrate of EGFR was investigated using LabChip (trademark) Systems (Caliper Life Sciences, Inc.). For t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2016
Entry Details
US Patent

TargetEpidermal growth factor receptor(Human)
Astellas Pharma

US Patent
LigandPNGBDBM170486(US9085540, 26)
Affinity DataIC50: 1.10nMAssay Description:The phosphorylation activity on the peptide substrate of EGFR was investigated using LabChip (trademark) Systems (Caliper Life Sciences, Inc.). For t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2016
Entry Details
US Patent