BDBM179711 US9127001, 8r::US9598410, Compound 8r

SMILES Fc1ccc(cc1)-c1nn(Cc2ccccc2)c2CCN(Cc12)C(=O)Cc1ccccc1

InChI Key InChIKey=ZYGQLOOEZVKRMO-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 179711   

TargetPotassium channel subfamily K member 3(Human)
Sanofi

US Patent
LigandPNGBDBM179711(US9127001, 8r | US9598410, Compound 8r)
Affinity DataIC50: 1.14E+3nMT: 2°CAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2016
Entry Details
US Patent

TargetPotassium channel subfamily K member 3(Human)
Sanofi

US Patent
LigandPNGBDBM179711(US9127001, 8r | US9598410, Compound 8r)
Affinity DataIC50: 1.14E+3nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent