BDBM192906 US9193689, IQ-157

SMILES Cc1cccc2c1cc([nH]c2=O)-c1cnc(nc1)N1CCN(CC1)C(=O)C1CC1

InChI Key InChIKey=QUSZOYLWBHWZLQ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 192906   

TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Human)
Institute of Cancer Research

US Patent
LigandPNGBDBM192906(US9193689, IQ-157)
Affinity DataIC50: 51nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2016
Entry Details
US Patent