BDBM195740 US9670212, 128 3-amino-N-[(2-{[2-(dimethylamino)ethyl](methyl)amino}-8-methylquinolin-3-yl)methyl]pyrazine-2-carboxamide

SMILES CN(C)CCN(C)c1nc2c(C)cccc2cc1CNC(=O)c1nccnc1N

InChI Key InChIKey=SUKJQIWWIVBIMW-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 195740   

LigandPNGBDBM195740(US9670212, 128 3-amino-N-[(2-{[2-(dimethylamino)et...)
Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent