BDBM195783 US9670212, 144 N-{[2-(4-ethylpiperazin-1-yl)-8-methylquinolin-3-yl]methyl}-9H-purin-6-amine

SMILES CCN1CCN(CC1)c1nc2c(C)cccc2cc1CNc1ncnc2[nH]cnc12

InChI Key InChIKey=YCCPKJXWSBFPKM-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 195783   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Exelixis

US Patent

LigandBDBM195783(US9670212, 144 N-{[2-(4-ethylpiperazin-1-yl)-8-met...)Copy SMILESCopy InChI

Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoKEGGPC cidPC sidSimilars

In Depth
Date in BDB:
7/7/2018
Entry Details
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