BDBM197741 US9216986, 2-[2-(6-Fluoro-quinolin-2-yl)-ethyl]-5-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-ol::US9801878, 2-[2-(6-Fluoro-quinolin-2-yl)-ethyl]-5-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-ol
SMILES Cc1ccc(O)c2nc(CCc3ccc4cc(F)ccc4n3)nn12
InChI Key InChIKey=SISLFPKXUFKGCB-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 197741
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Homo sapiens (Human))
H. Lundbeck
US Patent
H. Lundbeck
US Patent
Affinity DataIC50: 18nMAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A [440-779](Homo sapiens (Human))
H. Lundbeck
US Patent
H. Lundbeck
US Patent
Affinity DataIC50: 85nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair