BDBM202143 US9233983, I-14

SMILES CC1CN(Cc2ccc(nc2)-c2cc3c(ccnc3[nH]2)-c2cccc(N3CCOc4cc(cc(F)c4C3=O)C3CC3)c2CO)CC(C)N1C

InChI Key InChIKey=KLLDAQHHECGHJL-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 202143   

TargetTyrosine-protein kinase BTK(Human)
Advinus Therapeutics

US Patent
LigandPNGBDBM202143(US9233983, I-14)
Affinity DataIC50: 1.70nMAssay Description:The inhibition assays were performed using the generic tyrosine kinase assay kit from C is Bio (HTRF KinEASE-TK #62TK0PEB). The assay is based on the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2016
Entry Details
US Patent