BDBM204851 US9242977, 85-225

SMILES CCCNc1ncc(s1)-c1ccc(Oc2ncc(NC(=O)Nc3cc(ccc3S(=O)(=O)N(C)C)C(F)(F)F)cn2)cc1

InChI Key InChIKey=IVRDNDPVGALWJM-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 204851   

TargetIsoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)(Human)
Ono Pharmaceutical

US Patent

LigandBDBM204851(US9242977, 85-225)Copy SMILESCopy InChI

Affinity DataIC50: 4nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
12/6/2016
Entry Details
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