BDBM206001 1-(5-(4-((4-(5-((1R,3R)-2- (2,2-difluoroethyl)-3-methyl-2,3,4,9- tetrahydro-1H-pyrido[3,4-b]indol- 1-yl)pyrimidin-2-yl)piperazin-1- yl)methyl)piperidine-1-carbonyl)- 2-methoxyphenyl) dihydropyrimidine-2,4(1H,3H)-dione::US20260007681, Compound A7

SMILES COc1ccc(C(=O)N2CCC(CN3CCN(c4ncc([C@@H]5c6[nH]c7ccccc7c6C[C@@H](C)N5CC(F)F)cn4)CC3)CC2)cc1N1CCC(=O)NC1=O

InChI Key InChIKey=OMPNJRGJQFFFIQ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 206001   

TargetDNA damage-binding protein 1/Protein cereblon(Human)
University Of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 206001BDBM206001(1-(5-(4-((4-(5-((1R,3R)-2- (2,2-difluoroethyl)-3-m...)
Affinity DataIC50: 2.75E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2026
Entry Details
US Patent