BDBM225255 N-(2-phenyl-1-(3-phenylpropyl)-1H-benzo[d]imidazol-5-yl)-4-(trifluoromethoxy)benzenesulfonamide (16)

SMILES FC(F)(F)Oc1ccc(cc1)S(=O)(=O)Nc1ccc2n(CCCc3ccccc3)c(nc2c1)-c1ccccc1

InChI Key InChIKey=JQCQXEYYCPJVTQ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 225255   

TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225255(N-(2-phenyl-1-(3-phenylpropyl)-1H-benzo[d]imidazol...)
Affinity DataIC50: 2.19E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed