BDBM225256 4-Fluoro-N-(2-phenyl-1-(3-phenylpropyl)-1H-benzo[d]imidazol-5-yl)benzenesulfonamide (17)

SMILES Fc1ccc(cc1)S(=O)(=O)Nc1ccc2n(CCCc3ccccc3)c(nc2c1)-c1ccccc1

InChI Key InChIKey=BDVXUJQIADAYFH-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 225256   

TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225256(4-Fluoro-N-(2-phenyl-1-(3-phenylpropyl)-1H-benzo[d...)
Affinity DataIC50: 1.61E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed