BDBM250513 US9469639, Compound (VII)

SMILES Cc1ccc(F)c(NC(=O)Nc2ccc(-c3ccc(OCCC(C)(C)N)c4[nH]nc(N)c34)c3ccccc23)c1

InChI Key InChIKey=KRURSEZSUKLHMO-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 250513   

TargetVascular endothelial growth factor receptor 2(Human)
Radiant Pharma & Tech.

US Patent
LigandPNGBDBM250513(US9469639, Compound (VII))
Affinity DataIC50: 48.3nMT: 2°CAssay Description:Experimental Procedures(1) Kinase reaction substrate Poly(Glu, Tyr, 4:1) was diluted to 20 g/ml with potassium ion-free PBS, and enzyme labeled plate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
US Patent

TargetPlatelet-derived growth factor receptor beta(Human)
Radiant Pharma & Tech.

US Patent
LigandPNGBDBM250513(US9469639, Compound (VII))
Affinity DataIC50: 106nMT: 2°CAssay Description:Experimental Procedures(1) Kinase reaction substrate Poly(Glu, Tyr, 4:1) was diluted to 20 g/ml with potassium ion-free PBS, and enzyme labeled plate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
US Patent