BDBM255676 US9475815, 61

SMILES COc1cc(C)cc2cc(sc12)-c1cc(CNCC2CCN(C)CC2)n2ncnc(N)c12

InChI Key InChIKey=STKLVEJFSNEIDY-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 255676   

TargetFibroblast growth factor receptor 1 [400-80]/Glutathione S-transferase P(Human)
Bayer Intelletual Property

US Patent
LigandPNGBDBM255676(US9475815, 61)
Affinity DataIC50: 39.7nMpH: 7.0 T: 2°CAssay Description:A recombinant tagged FGFR-1 fusion protein [fusion of glutathione-S-transferase (GST) (N-terminally), His6-tag, thrombin cleavage site, and the intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 3 [397-806]/Glutathione S-transferase P(Human)
Bayer Intelletual Property

US Patent
LigandPNGBDBM255676(US9475815, 61)
Affinity DataIC50: 43.5nMpH: 7.0 T: 2°CAssay Description:A recombinant tagged FGFR-3 fusion protein [fusion of glutathione-S-transferase (GST) (N-terminally), His6-tag, thrombin cleavage site, and the intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2017
Entry Details
US Patent