BDBM256296 US9487488, 20

SMILES FC(F)(F)Oc1ccc(CN(c2ncc3ccccc3c2C(F)(F)F)S(=O)(=O)c2ccc(cc2)-c2ncn[nH]2)cc1

InChI Key InChIKey=DPJFLRCULAPHOA-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 256296   

TargetTransient receptor potential cation channel subfamily M member 8(Human)
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM256296(US9487488, 20)
Affinity DataIC50: 3.20nMT: 2°CAssay Description:The functional activity of a test compound was determined by measuring change in intracellular calcium concentration using a calcium sensitive fluore...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2017
Entry Details
US Patent