BDBM261768 Methyl 5-ethyl-5H-pyrido[3,2-b]indole-2-carboxylate::US9708311, 19

SMILES CCn1c2ccccc2c2nc(ccc12)C(=O)OC

InChI Key InChIKey=KUQKMCQSDUDHMJ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 261768   

TargetProstaglandin E2 receptor EP4 subtype(Human)
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM261768(Methyl 5-ethyl-5H-pyrido[3,2-b]indole-2-carboxylat...)
Affinity DataIC50: 32.2nMT: 2°CAssay Description:4 μl of a cAMP-d2/cell suspension (625000 cells/ml) were added to a test plate containing the substance solutions already initially introduced (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2018
Entry Details
US Patent