BDBM271142 7-(2,6-difluorobenzenesulfonyl)-2-methyl-4-(2-methylmorpholin-4-yl)-5H-pyrrolo[3,2-d]pyrimidin-6-amine::US10059713, Example 263

SMILES CC1CN(CCO1)c1nc(C)nc2c(c(N)[nH]c12)S(=O)(=O)c1c(F)cccc1F

InChI Key InChIKey=NSQNVRCLMOBDLR-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 271142   

TargetFree fatty acid receptor 2(Human)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM271142(7-(2,6-difluorobenzenesulfonyl)-2-methyl-4-(2-meth...)
Affinity DataEC50:  5nMAssay Description:GPR43 agonist/PAM activity was determined by measuring changes in intracellular calcium levels using a Ca2+ sensitive fluorescent dye. The changes in...More data for this Ligand-Target Pair
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Date in BDB:
12/11/2018
Entry Details
US Patent