BDBM2713 3-[6,7,8,9-Tetrahydro-8-[(trimethylamino)methyl]pyrido[1,2-a]indol-10-yl]-4-(1-methyl-3-indolyl)-1H-pyrrole-2,5-dione Trifluoromethanesulfonate::Bisindolylmaleimide deriv. 18c::trimethyl({10-[4-(1-methyl-1H-indol-3-yl)-2,5-dioxo-2,5-dihydro-1H-pyrrol-3-yl]-1H,2H,3H,4H-pyrido[1,2-a]indol-2-yl}methyl)azanium

SMILES Cn1cc(C2=C(C(=O)NC2=O)c2c3CC(C[N+](C)(C)C)CCn3c3ccccc23)c2ccccc12

InChI Key InChIKey=ACDXNHQLUBRPFY-UHFFFAOYSA-O

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 2713   

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2713(3-[6,7,8,9-Tetrahydro-8-[(trimethylamino)methyl]py...)
Affinity DataIC50: 49nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2004
Entry Details Article
PubMed
LigandPNGBDBM2713(3-[6,7,8,9-Tetrahydro-8-[(trimethylamino)methyl]py...)
Affinity DataIC50: 9.25E+4nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2004
Entry Details Article
PubMed