BDBM278624 (2E)-[1-({5-[1- (Methylamino)cyclopropyl]-3- (2,4,6-trichlorophenyl)-1,2- oxazol-4-yl}carbonyl)-3,4- dihydrobenzo[cd]indol-5(1H)- ylidene]ethanoic acid ::US10040791, Example 86
SMILES CNC1(CC1)c1onc(c1C(=O)n1cc2CC\C(=C/C(O)=O)c3cccc1c23)-c1c(Cl)cc(Cl)cc1Cl
InChI Key InChIKey=VOQZIABIIAPGMT-UKTHLTGXSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 278624
Affinity DataIC50: 79nMpH: 7.5 T: 25°CAssay Description:The IDH1R132H protein and the IDH1R132C protein were prepared as follows: the IDH1R132H or IDH1R132C gene was integrated into a pET24b(+) vector (Nov...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMpH: 7.5 T: 25°CAssay Description:The IDH1R132H protein and the IDH1R132C protein were prepared as follows: the IDH1R132H or IDH1R132C gene was integrated into a pET24b(+) vector (Nov...More data for this Ligand-Target Pair