BDBM280371 US10030012, Example 1::ethyl 4-[4- (1-methyl- 1H-imidazol- 2-yl)piperidin-1- yl]piperidine- 1-carboxylate

SMILES CCOC(=O)N1CCC(CC1)N1CCC(CC1)c1nccn1C

InChI Key InChIKey=WNWACNMKTQFVQH-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 280371   

TargetMuscarinic acetylcholine receptor M4(Human)
Heptares Therapeutics

US Patent
LigandPNGBDBM280371(ethyl 4-[4- (1-methyl- 1H-imidazol- 2-yl)piperidin...)
Affinity DataEC50:  2.36E+3nMAssay Description:The functional activity of compounds at the M4 and M2 receptors was determined by measuring changes in the level of intracellular calcium ions caused...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M2(Human)
Heptares Therapeutics

US Patent
LigandPNGBDBM280371(ethyl 4-[4- (1-methyl- 1H-imidazol- 2-yl)piperidin...)
Affinity DataEC50: >1.00E+7nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2018
Entry Details
US Patent