BDBM280409 US10030012, Example 39::ethyl 4-[4-(1- methyl-2-oxo-1,2- dihydropyridin-3- yl)piperidin-1- yl]azepane-1- carboxylate

SMILES CCOC(=O)N1CCCC(CC1)N1CCC(CC1)c1cccn(C)c1=O

InChI Key InChIKey=MQBKISVAZIHSRI-UHFFFAOYSA-N

Data  1 EC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 280409   

TargetMuscarinic acetylcholine receptor M4(Human)
Heptares Therapeutics

US Patent
LigandPNGBDBM280409(ethyl 4-[4-(1- methyl-2-oxo-1,2- dihydropyridin-3-...)
Affinity DataEC50:  740nMAssay Description:The functional activity of compounds at the M4 and M2 receptors was determined by measuring changes in the level of intracellular calcium ions caused...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2018
Entry Details
US Patent