BDBM286729 6-Bromo-3-(5- chloro-2- ethanesulfonyl- benzyl)-7-((R)-3- methylamino- piperidin-1- ylmethyl)-1H- quinazoline-2,4- dione::US9567304, Compound E-17

SMILES CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCC[C@H](C3)NC)c(Br)cc2c1=O

InChI Key InChIKey=ISNZQSZUBPYOQH-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 286729   

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandPNGBDBM286729(6-Bromo-3-(5- chloro-2- ethanesulfonyl- benzyl)-7-...)
Affinity DataIC50: 20nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent