BDBM28689 2-({3-[(6-chloro-1H-indole-1-)sulfonyl]benzene}amido)-5-methylbenzoic acid::Anthranilic acid deriv., 27

SMILES Cc1ccc(NC(=O)c2cccc(c2)S(=O)(=O)n2ccc3ccc(Cl)cc23)c(c1)C(O)=O

InChI Key InChIKey=ATXPCFTUFHGWSH-UHFFFAOYSA-N

Data  6 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 28689   

TargetPeroxisome proliferator-activated receptor delta(Human)
Universidad Nacional Aut£Noma De M£Xico

Curated by ChEMBL
LigandPNGBDBM28689(2-({3-[(6-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50: 63.0nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Universidad Nacional Aut£Noma De M£Xico

Curated by ChEMBL
LigandPNGBDBM28689(2-({3-[(6-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50: 63nM EC50:  200nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28689(2-({3-[(6-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50: 2.00E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28689(2-({3-[(6-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50: 2.00E+3nMAssay Description:Agonist activity at PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
LigandPNGBDBM28689(2-({3-[(6-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50: 3.16E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28689(2-({3-[(6-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50: 3.16E+3nMAssay Description:Agonist activity at PPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed