BDBM293967 US10106552, Compound 42

SMILES NC(=O)c1sc2nc3c(CCCC33CCCC3)c(-c3cncs3)c2c1N

InChI Key InChIKey=VYPVYMABMMIJQM-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 293967   

TargetEukaryotic elongation factor 2 kinase(Human)
Longevica Pharmaceuticals

US Patent
LigandPNGBDBM293967(US10106552, Compound 42)
Affinity DataIC50: 3.10E+3nMAssay Description:To determine the IC50 of compounds of the invention, recombinant eEF2K was diluted in an assay buffer in the presence of calmodulin, a calcium-bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent