BDBM294019 (2S)-5-((4-(1-(1H-Tetrazol-5- yl)pent-3-yn-2- yl)phenoxy)methyl)-3-(2- methylphenyl)thieno[2,3- c]pyridine::US10106553, Compound 51

SMILES CC#C[C@@H](Cc1nnn[nH]1)c1ccc(OCc2cc3c(csc3cn2)-c2ccccc2C)cc1

InChI Key InChIKey=UBKBYXJMQMWQPI-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 294019   

TargetFree fatty acid receptor 1(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM294019(US10106553, Compound 51 | (2S)-5-((4-(1-(1H-Tetraz...)
Affinity DataEC50:  3nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent