BDBM296168 2-[1-(oxan-4-yl)indol-5-yl]oxypyrido[3,4- d]pyrimidin-4-ol::US10112940, Example 91::US10202381, Example 91::US10208039, Example 91::US10611763, Example 91::US10815234, Example 91::US11535616, Example 91

SMILES Oc1nc(Oc2ccc3n(ccc3c2)C2CCOCC2)nc2cnccc12

InChI Key InChIKey=LPQYVJZVLPGAOE-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 296168   

TargetLysine-specific demethylase 4C(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM296168(US10112940, Example 91 | 2-[1-(oxan-4-yl)indol-5-y...)
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2019
Entry Details
US Patent

TargetLysine-specific demethylase 4C(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM296168(US10112940, Example 91 | 2-[1-(oxan-4-yl)indol-5-y...)
Affinity DataIC50: 550nMAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate-format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent