BDBM296173 2-[4-(3-fluoro-N- methylanilino)phenoxy]pyrido[3,4- d]pyrimidin-4-ol::US10112940, Example 96::US10202381, Example 96::US10208039, Example 96::US10611763, Example 96::US10815234, Example 96::US11535616, Example 96

SMILES CN(c1ccc(Oc2nc(O)c3ccncc3n2)cc1)c1ccccc1F

InChI Key InChIKey=GGHUFCYASQYURN-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 296173   

TargetLysine-specific demethylase 4C(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM296173(US10112940, Example 96 | 2-[4-(3-fluoro-N- methyla...)
Affinity DataIC50: 550nMAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate-format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetLysine-specific demethylase 4C(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM296173(US10112940, Example 96 | 2-[4-(3-fluoro-N- methyla...)
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2019
Entry Details
US Patent