BDBM296176 2-[4-[N-methyl-4-(oxan-4- yl)anilino]phenoxy]pyrido[3,4-d]pyrimidin- 4-ol::US10112940, Example 99::US10202381, Example 99::US10208039, Example 99::US10611763, Example 99::US10815234, Example 99::US11535616, Example 99

SMILES CN(c1ccc(Oc2nc(O)c3ccncc3n2)cc1)c1ccc(cc1)C1CCOCC1

InChI Key InChIKey=BLJSTINEDBDJEQ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 296176   

TargetLysine-specific demethylase 4C(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM296176(US10112940, Example 99 | 2-[4-[N-methyl-4-(oxan-4-...)
Affinity DataIC50: 550nMAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate-format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetLysine-specific demethylase 4C(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM296176(US10112940, Example 99 | 2-[4-[N-methyl-4-(oxan-4-...)
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2019
Entry Details
US Patent