BDBM297434 4-({[6-Bromo-3-methyl-2-(2-methylphenyl)quinolin-4-yl]carbonyl}amino)bicyclo[2.2.2]octane-1-carboxylic acid::US10117864, Example 24

SMILES Cc1ccccc1-c1nc2ccc(Br)cc2c(C(=O)NC23CCC(CC2)(CC3)C(O)=O)c1C

InChI Key InChIKey=QJNARVCAJMPGFR-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 297434   

TargetProstaglandin F2-alpha receptor(Human)
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM297434(US10117864, Example 24 | 4-({[6-Bromo-3-methyl-2-(...)
Affinity DataIC50: 129nMAssay Description:For the characterization of test substances in respect of FP antagonism, PGF2α-induced calcium flux in FP-expressing CHEM1 cells (Millipore, HTS...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
US Patent