BDBM298388 US10124003, Ex. Compound 69

SMILES COc1cc(OC)cc(c1)C#Cc1cn([C@@H]2C[C@@H](N(C2)C(=O)C=C)c2nnc(C)o2)c2ncnc(N)c12

InChI Key InChIKey=UQJJVELGKQUUJN-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 298388   

TargetFibroblast growth factor receptor 2(Human)
Taiho Pharmaceutical

US Patent
LigandPNGBDBM298388(US10124003, Ex. Compound 69)
Affinity DataIC50: 8.80nMAssay Description:When setting conditions for the measurement of the inhibitory effect of the compounds on FGFR2 kinase activity, FL-Peptide 22 (Caliper Life Sciences,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
US Patent