BDBM30004 benzimidazole analogue, 7c

SMILES CCOC(=O)N1CCC(C)(CC1)Sc1nc2cc(Cl)c(cc2[nH]1)N1CCN(CC)CC1

InChI Key InChIKey=ZUPHLBSFYJTEQV-UHFFFAOYSA-N

Data  2 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 30004   

TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM30004(benzimidazole analogue, 7c)
Affinity DataIC50: 4.30nM EC50:  1.10nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM30004(benzimidazole analogue, 7c)
Affinity DataIC50: 3.90E+3nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed