BDBM316183 N-(4-methoxy-3-nitrophenyl)-6-(2-methoxyphenyl)pyrimidin-4-amine::US10294218, Example 11::US9617225, Example 11

SMILES COc1ccccc1-c1cc(Nc2ccc(OC)c(c2)[N+]([O-])=O)ncn1

InChI Key InChIKey=ZHFNQFDJLZJRPE-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 316183   

TargetCyclin-dependent kinase 9(Human)
Virostatics

US Patent
LigandPNGBDBM316183(US9617225, Example 11 | N-(4-methoxy-3-nitrophenyl...)
Affinity DataIC50: 1.00E+3nMAssay Description:The activity of the compounds described in the present invention can be determined by measuring the phosphorylation of a fluorescently-labeled peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Virostatics

US Patent
LigandPNGBDBM316183(US9617225, Example 11 | N-(4-methoxy-3-nitrophenyl...)
Affinity DataIC50: 1.00E+3nMAssay Description:The activity of the compounds described in the present invention can be determined by measuring the phosphorylation of a fluorescently-labeled peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetCyclin-dependent kinase 9(Human)
Virostatics

US Patent
LigandPNGBDBM316183(US9617225, Example 11 | N-(4-methoxy-3-nitrophenyl...)
Affinity DataIC50: 1.00E+3nMAssay Description:The activity of the compounds described in the present invention can be determined by measuring the phosphorylation of a fluorescently-labeled peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Virostatics

US Patent
LigandPNGBDBM316183(US9617225, Example 11 | N-(4-methoxy-3-nitrophenyl...)
Affinity DataIC50: 1.00E+3nMAssay Description:The activity of the compounds described in the present invention can be determined by measuring the phosphorylation of a fluorescently-labeled peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent