BDBM318021 8-Methyl-2-[4-[[5-trifluoromethyl)pyrimidin-2- yl]methyl)piperazin-1-yl]- 3,5,6,7-tetrahydropyrido[2,3- d]pyrimidin-4-one::US9624218, Example 15
SMILES CN1CCCc2c1nc([nH]c2=O)N1CCN(Cc2ncc(cn2)C(F)(F)F)CC1
InChI Key InChIKey=DTOVAHAAYGWZJC-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 318021
Affinity DataIC50: 25.3nMAssay Description:The enzymatic activity of hTNKS1 and hTNKS2 is assessed using an enzyme-linked immunosorbent assay (ELISA) which detects poly ADP ribose incorporated...More data for this Ligand-Target Pair
Affinity DataIC50: 6.91E+3nMAssay Description:The Poly ADP-ribose polymerase 1(PARP1) assay is an ELISA which detects poly ADP ribose incorporated into plate-bound histone protein in a 384-well f...More data for this Ligand-Target Pair
Affinity DataIC50: 16.7nMAssay Description:The enzymatic activity of hTNKS1 and hTNKS2 is assessed using an enzyme-linked immunosorbent assay (ELISA) which detects poly ADP ribose incorporated...More data for this Ligand-Target Pair