BDBM318919 1-methyl-6-(2-(2,2,2-trifluoroethoxy)phenyl)-1H-indazol-3-amine::US10173985, Example 8

SMILES Cn1nc(N)c2ccc(cc12)-c1ccccc1OCC(F)(F)F

InChI Key InChIKey=QJVJMKKSESPJFR-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 318919   

TargetSodium channel protein type 9 subunit alpha(Human)
Almirall

US Patent
LigandPNGBDBM318919(US10173985, Example 8 | 1-methyl-6-(2-(2,2,2-trifl...)
Affinity DataIC50: 320nMAssay Description:Electrophysiological studies are performed with an IonWorks Quattro (Molecular Devices Corp.) automated patch-clamp electrophysiology platform as des...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetSodium channel protein type 5 subunit alpha(Human)
Almirall

US Patent
LigandPNGBDBM318919(US10173985, Example 8 | 1-methyl-6-(2-(2,2,2-trifl...)
Affinity DataIC50: 3.30E+4nMAssay Description:Electrophysiological studies are performed with an IonWorks Quattro (Molecular Devices Corp.) automated patch-clamp electrophysiology platform as des...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent