BDBM323253 (S)-N-[(R)-2-(3-Butoxy-3-o-tolylazetidin-1-yl)-1-(4-methoxybenzyl)-2-oxoethyl]-2-hydroxy-3-(1H-imidazol-4-yl)propionamide::US9630949, 71

SMILES CCCCOC1(CN(C1)C(=O)[C@@H](Cc1ccc(OC)cc1)NC(=O)[C@@H](O)Cc1c[nH]cn1)c1ccccc1C

InChI Key InChIKey=WDKZSCBDFMWRDB-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 323253   

TargetMelanocyte-stimulating hormone receptor(Human)
Galderma Research & Development

US Patent
LigandPNGBDBM323253((S)-N-[(R)-2-(3-Butoxy-3-o-tolylazetidin-1-yl)-1-(...)
Affinity DataEC50:  60nMAssay Description:In the presence of an activator (agonist), the melanocortin receptor will activate the cAMP pathway which, via the CRE-Luc vector, will result in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2019
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Galderma Research & Development

US Patent
LigandPNGBDBM323253((S)-N-[(R)-2-(3-Butoxy-3-o-tolylazetidin-1-yl)-1-(...)
Affinity DataEC50:  4.00E+3nMAssay Description:In the presence of an activator (agonist), the melanocortin receptor will activate the cAMP pathway which, via the CRE-Luc vector, will result in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2019
Entry Details
US Patent