BDBM3245 (3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl 4-{[2-(butoxycarbonyl)-6-hydroxyphenyl]carbonyl}-3,5-dihydroxybenzoate::Balanol Benzophenone Ester Analog 17

SMILES CCCCOC(=O)c1cccc(O)c1C(=O)c1c(O)cc(cc1O)C(=O)O[C@@H]1CNC[C@H]1NC(=O)c1ccc(O)cc1

InChI Key InChIKey=NXOILRDXHDPZAY-UHFFFAOYSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 3245   

TargetProtein kinase C eta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3245((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 40nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C delta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3245((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 80nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C beta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3245((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 2.20E+3nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C alpha type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3245((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 3.10E+3nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C epsilon type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3245((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 3.70E+3nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article