BDBM32471 piperazine amide, 4r

SMILES Brc1ccc(o1)C(=O)Nc1cccc(Br)c1N1CCN(CC=C)CC1

InChI Key InChIKey=KRMXSKGWRKZWPH-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 32471   

TargetMitogen-activated protein kinase 8(Human)
The Scripps Research Institute

LigandPNGBDBM32471(piperazine amide, 4r)
Affinity DataIC50: 2.00E+4nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandPNGBDBM32471(piperazine amide, 4r)
Affinity DataIC50: 2.00E+4nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed