BDBM329171 4-(5-chloro-6-((1R)-1-(2,5-dichlorophenyl)ethoxy)-3-pyridinyl)-2-fluoro-5-methyl-N-(methylsulfonyl)benzamide::US9663508, Example 673

SMILES C[C@@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O)c1cc(Cl)ccc1Cl

InChI Key InChIKey=AIJTXLAXVVHOOZ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 329171   

LigandPNGBDBM329171(US9663508, Example 673 | 4-(5-chloro-6-((1R)-1-(2,...)
Affinity DataIC50: 46.2nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandPNGBDBM329171(US9663508, Example 673 | 4-(5-chloro-6-((1R)-1-(2,...)
Affinity DataIC50: 1.00E+4nMAssay Description:293 cells stably transfected with human Nav 1.5 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology syste...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent