BDBM331954 6-(2,3-dichlorophenyl)-N3-(2-((2-(2-methoxyethoxy)ethyl)(methyl)amino)ethyl)-N3-methyl-1,2,4-triazine-3,5-diamine ::US10189859, Compound 193

SMILES COCCOCCN(C)CCN(C)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl

InChI Key InChIKey=QBVYPFKFOJQOTE-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 331954   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Nektar Therapeutics

US Patent
LigandPNGBDBM331954(6-(2,3-dichlorophenyl)-N3-(2-((2-(2-methoxyethoxy)...)
Affinity DataIC50: <5.00E+4nMAssay Description:The potencies of the compounds provided herein to block specific Na+ channels was measured using automated patch clamp electrophysiologically of Nav1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Nektar Therapeutics

US Patent
LigandPNGBDBM331954(6-(2,3-dichlorophenyl)-N3-(2-((2-(2-methoxyethoxy)...)
Affinity DataIC50:  6.26E+4nMAssay Description:The potencies of the compounds provided herein to block specific Na+ channels was measured using automated patch clamp electrophysiologically of Nav1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent