BDBM355727 US9815820, Y-27263

SMILES CC(C)[C@H]1CC[C@@H](CC1)C(=O)Nc1ccncc1

InChI Key InChIKey=ZOJWMHJRZRKSRN-UHFFFAOYSA-N

Data  2 KI  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 355727   

TargetRho-associated protein kinase 1(Human)
Kadmon

US Patent
LigandPNGBDBM355727(US9815820, Y-27263)
Affinity DataKi:  40nMAssay Description:Kinase inhibition can be determined using an IMAP assay (Molecular Devices). This assay method involves the use of a fluorescently-tagged peptide sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2019
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandPNGBDBM355727(US9815820, Y-27263)
Affinity DataKi:  60nMAssay Description:Kinase inhibition can be determined using an IMAP assay (Molecular Devices). This assay method involves the use of a fluorescently-tagged peptide sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2019
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Kadmon

US Patent
LigandPNGBDBM355727(US9815820, Y-27263)
Affinity DataIC50: 1.13E+3nMAssay Description:Kinase inhibition can be determined using an IMAP assay (Molecular Devices). This assay method involves the use of a fluorescently-tagged peptide sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2019
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandPNGBDBM355727(US9815820, Y-27263)
Affinity DataIC50: 1.63E+3nMAssay Description:Kinase inhibition can be determined using an IMAP assay (Molecular Devices). This assay method involves the use of a fluorescently-tagged peptide sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2019
Entry Details
US Patent