BDBM362930 US9849138, 4
SMILES CN1c2ccccc2C(=O)NC(Cc2ccc(cc2)-c2ccncc2)C1=O
InChI Key InChIKey=LJOQPYLDIOBLQD-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 362930
TargetRho-associated protein kinase 2 [11-552](Human)
The Regents of The University of Michigan
US Patent
The Regents of The University of Michigan
US Patent
Affinity DataIC50: 800nMAssay Description:In a final reaction volume of 25 μL, ROCK-II (h, amino acids 11-552) (5-10 mU) was incubated with 50 mM Tris pH 7.5, 0.1 mM EGTA, 30 μM KEA...More data for this Ligand-Target Pair
TargetRho-associated protein kinase 1 [17-535](Human)
The Regents of The University of Michigan
US Patent
The Regents of The University of Michigan
US Patent
Affinity DataIC50: >1.00E+7nMAssay Description:In a final reaction volume of 25 μL, ROCK-I (h, amino acids 17-535) (5-10 mU) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 μM KEAKE...More data for this Ligand-Target Pair