BDBM369254 N-[(4-fluorophenyl)methyl]-4-[6-(1- methylsulfonyl-3,6-dihydro-2H-pyridin-4- yl)thieno[3,2-d]pyrimidin-4-yl]piperazine- 1-carboxamide::US10227357, Compound P-0568
SMILES CS(=O)(=O)N1CCC(=CC1)c1cc2ncnc(N3CCN(CC3)C(=O)NCc3ccc(F)cc3)c2s1
InChI Key InChIKey=LHMWQPDWCWXZJM-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 369254
Affinity DataKi: 500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Affinity DataKi: 5.50E+3nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair