BDBM369503 N-[2-[4-[[(1R,2S)-2-phenylcyclopropyl]amino]-1-piperidyl]propyl]methanesulfonamide::US10233152, Example 41

SMILES CC(CNS(C)(=O)=O)N1CCC(CC1)N[C@@H]1C[C@H]1c1ccccc1

InChI Key InChIKey=VHLYSAMXJQKDAV-UHFFFAOYSA-N

Data  1 IC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 369503   

TargetLysine-specific histone demethylase 1A(Human)
Mirati Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 369503BDBM369503(N-[2-[4-[[(1R,2S)-2-phenylcyclopropyl]amino]-1-pip...)
Affinity DataIC50: 15nMAssay Description:Briefly, compounds of the present invention were solubilized in DMSO and a series of 10, three-fold serial dilutions were made for each compound in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2019
Entry Details
US Patent